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Molecular modeling and evaluation of binding mode and affinity of artemisinin-quinine hybrid and its congeners with Fe-protoporphyrin-IX as a putative receptor

A recent rational approach to anti-malarial drug design is characterized as “covalent biotherapy” involves linking of two molecules with individual intrinsic activity into a single agent, thus packaging dual activity into a single hybrid molecule. In view of this background and reported anti malaria...

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Autori principali: Mahapatra, Rajani Kanta, Behera, Niranjan, Naik, Pradeep Kumar
Natura: Artigo
Lingua:Inglês
Pubblicazione: Biomedical Informatics 2012
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3346024/
https://ncbi.nlm.nih.gov/pubmed/22570518
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.6026/97320630008369
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