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Libraries of 2,3,4,6,7,11b-Hexahydro-1H-pyrido[2,1-a]isoquinolin-2-amine Derivatives via a Multicomponent Assembly Process/1,3-Dipolar Cycloaddition Strategy

A Mannich-type multicomponent assembly process/1,3-dipolar cycloaddition strategy has been developed for the rapid and efficient construction of a parent tetrahydroisoquinoline fused isoxazolidine scaffold, which was subsequently functionalized using well-established protocols to access a diverse 70...

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Detalhes bibliográficos
Main Authors: Granger, Brett A., Kaneda, Kyosuke, Martin, Stephen F.
Formato: Artigo
Idioma:Inglês
Publicado em: 2011
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3253940/
https://ncbi.nlm.nih.gov/pubmed/22040015
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/co2001636
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