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Antitrypanosomal Activity of Fexinidazole, a New Oral Nitroimidazole Drug Candidate for Treatment of Sleeping Sickness

Fexinidazole is a 5-nitroimidazole drug currently in clinical development for the treatment of human sleeping sickness (human African trypanosomiasis [HAT]), caused by infection with species of the protozoan parasite Trypanosoma brucei. The compound and its two principal metabolites, sulfoxide and s...

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Autori principali: Kaiser, Marcel, Bray, Michael A., Cal, Monica, Bourdin Trunz, Bernadette, Torreele, Els, Brun, Reto
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Society for Microbiology 2011
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3232772/
https://ncbi.nlm.nih.gov/pubmed/21911566
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.00246-11
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