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Homology modeling of mosquito cytochrome P450 enzymes involved in pyrethroid metabolism: insights into differences in substrate selectivity

BACKGROUND: Cytochrome P450 enzymes (P450s) have been implicated in insecticide resistance. Anopheles minumus mosquito P450 isoforms CYP6AA3 and CYP6P7 are capable of metabolizing pyrethroid insecticides, however CYP6P8 lacks activity against this class of compounds. FINDINGS: Homology models of the...

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Autori principali: Lertkiatmongkol, Panida, Jenwitheesuk, Ekachai, Rongnoparut, Pornpimol
Natura: Artigo
Lingua:Inglês
Pubblicazione: BioMed Central 2011
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3228512/
https://ncbi.nlm.nih.gov/pubmed/21892968
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1186/1756-0500-4-321
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