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Sex Difference in κ-Opioid Receptor (KOPR)-Mediated Behaviors, Brain Region KOPR Level and KOPR-Mediated Guanosine 5′-O-(3-[(35)S]Thiotriphosphate) Binding in the Guinea Pig

We examined whether sex differences in κ-opioid receptor (KOPR) pharmacology exist in guinea pigs, which are more similar to humans in the expression level and distribution of KOPR in the brain than rats and mice. The KOPR agonist trans-(±)-3,4-dichloro-N-methyl-N-(2-[1-pyrrolidinyl]-cyclohexyl)benz...

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Autors principals: Wang, Yu-Jun, Rasakham, Khampaseuth, Huang, Peng, Chudnovskaya, Darina, Cowan, Alan, Liu-Chen, Lee-Yuan
Format: Artigo
Idioma:Inglês
Publicat: The American Society for Pharmacology and Experimental Therapeutics 2011
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3199977/
https://ncbi.nlm.nih.gov/pubmed/21841040
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/jpet.111.183905
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