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Phase I study of continuous MKC-1 in patients with advanced or metastatic solid malignancies using the modified Time-to-Event Continual Reassessment Method (TITE-CRM) dose escalation design

BACKGROUND: MKC-1 is an oral cell-cycle inhibitor with broad antitumor activity in preclinical models. Clinical studies demonstrated modest antitumor activity using intermittent dosing schedule, however additional preclinical data suggested continuous dosing could be efficacious with additional effe...

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Detalhes bibliográficos
Main Authors: Tevaarwerk, Amye, Wilding, George, Eickhoff, Jens, Chappell, Rick, Sidor, Carolyn, Arnott, Jamie, Bailey, Howard, Schelman, William, Liu, Glenn
Formato: Artigo
Idioma:Inglês
Publicado em: 2011
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3139017/
https://ncbi.nlm.nih.gov/pubmed/21225315
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s10637-010-9629-6
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