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Small molecule inhibitors of SHP2 tyrosine phosphatase discovered by virtual screening

SHP2, encoded by PTPN11, is a non-receptor protein tyrosine phosphatase (PTP) containing two tandem Src homology-2 (SH2) domains. It is expressed ubiquitously and plays critical roles in growth factor mediated processes, primarily by promoting the activation of the RAS/ERK signaling pathway. Genetic...

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Библиографические подробности
Главные авторы: Yu, Zhi-Hong, Chen, Lan, Wu, Li, Liu, Sijiu, Wang, Lina, Zhang, Zhong-Yin
Формат: Artigo
Язык:Inglês
Опубликовано: 2011
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC3128679/
https://ncbi.nlm.nih.gov/pubmed/21669525
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2011.05.078
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