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A UPLC-MS/MS assay of the “Pittsburgh Cocktail”: six CYP probe-drug/metabolites from human plasma and urine using stable isotope dilution

The efficiency of drug metabolism by a single enzyme can be measured as the fractional metabolic clearance which can be used as a measure of whole body activity for that enzyme. Measurement of activity of multiple enzymes simultaneously is feasible using a cocktail approach however analytical approa...

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Autores principales: Stewart, Nicolas A., Buch, Shama C., Conrads, Thomas P., Branch, Robert A.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2010
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC3115584/
https://ncbi.nlm.nih.gov/pubmed/21107456
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c0an00643b
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