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The diterpenoid alkaloid noroxoaconitine is a Mapkap kinase 5 (MK5/PRAK) inhibitor

The mitogen-activated protein kinase-activated protein kinase MK5 is ubiquitously expressed in vertebrates and is implicated in cell proliferation, cytoskeletal remodeling, and anxiety behavior. This makes MK5 an attractive drug target. We tested several diterpenoid alkaloids for their ability to su...

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Bibliografski detalji
Glavni autori: Kostenko, Sergiy, Khan, Mahmud Tareq Hassan, Sylte, Ingebrigt, Moens, Ugo
Format: Artigo
Jezik:Inglês
Izdano: SP Birkhäuser Verlag Basel 2010
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3016492/
https://ncbi.nlm.nih.gov/pubmed/20640477
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s00018-010-0452-1
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