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In Silico-Experimental Approach for Drug Design: the Binding Mode of Peptidic and Non Peptidic Inhibitors to Hsp90 N-Terminal Domain

Heat shock protein 90 (Hsp90) is a prime target for antitumor therapies. The information obtained by MD simulations is combined with NMR data to provide a cross-validated atomic resolution model of the complementary interactions of Hsp90 with a peptidic (Shepherdin) and a non peptidic (5-aminoimidaz...

पूर्ण विवरण

में बचाया:
ग्रंथसूची विवरण
मुख्य लेखकों: Tomaselli, Simona, Meli, Massimiliano, Plescia, Janet, Zetta, Lucia, Altieri, Dario C., Colombo, Giorgio, Ragona, Laura
स्वरूप: Artigo
भाषा:Inglês
प्रकाशित: 2010
विषय:
ऑनलाइन पहुंच:https://ncbi.nlm.nih.gov/pmc/articles/PMC2953720/
https://ncbi.nlm.nih.gov/pubmed/20925690
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/j.1747-0285.2010.01015.x
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