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Gabapentin suppresses cortical spreading depression susceptibility

Cortical spreading depression (CSD) is an intense depolarization wave implicated in the pathophysiology of brain injury states and migraine aura. As Ca(v)2.1 channels modulate CSD susceptibility, we tested gabapentin, which inhibits Ca(v)2.1 through high-affinity binding to its α(2)δ subunit, on CSD...

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Detalhes bibliográficos
Main Authors: Hoffmann, Ulrike, Dileköz, Ergin, Kudo, Chiho, Ayata, Cenk
Formato: Artigo
Idioma:Inglês
Publicado em: Nature Publishing Group 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2949257/
https://ncbi.nlm.nih.gov/pubmed/20588320
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/jcbfm.2010.92
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