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Diminished sensitivity of Chronic Lymphocytic Leukemia cells to ABT-737 and ABT-263 due to albumin binding in blood

PURPOSE: Inhibition of the anti-apoptotic BCL2 family is one of the most promising areas of anti-cancer drug development. However, ABT-737, a specific BCL2 inhibitor, is neither orally bioavailable nor metabolically stable. To overcome these problems, the structurally related molecule, ABT-263, was...

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Библиографические подробности
Главные авторы: Vogler, Meike, Furdas, Silviya D, Jung, Manfred, Kuwana, Tomomi, Dyer, Martin JS, Cohen, Gerald M
Формат: Artigo
Язык:Inglês
Опубликовано: 2010
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC2921948/
https://ncbi.nlm.nih.gov/pubmed/20601444
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/1078-0432.CCR-10-0777
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