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In Vitro Structure-Activity Relationship of Re-cyclized Octreotide Analogues

INTRODUCTION: Development of radiolabeled octreotide analogues is of interest for targeting somatostatin receptor-positive tumors for diagnostic and therapeutic purposes. We are investigating a direct labeling approach for incorporation of a Re ion into octreotide analogues, where the peptide sequen...

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Detalles Bibliográficos
Autores principales: Dannoon, Shorouk F., Bigott-Hennkens, Heather M., Ma, Lixin, Gallazzi, Fabio, Lewis, Michael R., Jurisson, Silvia S.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2010
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC2901243/
https://ncbi.nlm.nih.gov/pubmed/20610157
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.nucmedbio.2010.03.008
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