Caricamento...

Potent and use-dependent block of cardiac sodium channels by U-50,488H, a benzeneacetamide kappa opioid receptor agonist

OBJECTIVES: To determine whether the kappa opioid receptor agonist U-50,488H, a benzacetamide derivative of the cyclo-hexane-1,2-diamine analgesics, may be a useful molecular probe to define the structural requirements of this class of drugs for cardiac sodium channel blockade. ANIMALS AND METHODS:...

Descrizione completa

Salvato in:
Dettagli Bibliografici
Autori principali: Pugsley, Michael K, Yu, Esther J, Goldin, Alan L
Natura: Artigo
Lingua:Inglês
Pubblicazione: Pulsus Group Inc 2001
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2859007/
https://ncbi.nlm.nih.gov/pubmed/20428265
Tags: Aggiungi Tag
Nessun Tag, puoi essere il primo ad aggiungerne! !