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Quaternary ammonium compounds efficiently inhibit Plasmodium falciparum growth in vitro by impairment of choline transport.

Hemicholinium 3, decamethonium, and decyltrimethylammonium previously have been demonstrated to be efficient inhibitors, with 50% inhibitory concentrations of 4 X 10(-6), 10(-6), and 7 X 10(-7) M, respectively. We show that lengthening of the alkyl chain of decyltrimethylammonium by successive addit...

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Detalhes bibliográficos
Publicado no:Antimicrob Agents Chemother
Principais autores: Ancelin, M L, Vial, H J
Formato: Artigo
Idioma:Inglês
Publicado em: American Society for Microbiology (ASM) 1986
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.govhttps://pmc.ncbi.nlm.nih.gov/articles/PMC284159/
https://ncbi.nlm.nih.govhttps://pubmed.ncbi.nlm.nih.gov/3524430/
https://ncbi.nlm.nih.govhttps://doi.org/10.1128/aac.29.5.814
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