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3ircular dichroism simulation shows a site-II-to-site-I displacement of human serum albumin-bound diclofenac by ibuprofen

Purpose: The purpose of this study was to confirm the hypothesis that a site-II-to-site-I displacement takes place when some nonsteroidal anti-inflammatory drugs are displaced by another drug from their high-affinity binding site to a site of lower affinity on human serum albumin (HSA).Methods: Dicl...

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Detalhes bibliográficos
Main Authors: Yamasaki, Keishi, Rahman, Mohammed Hablbur, Tsutsumi, Yasuhiro, Maruyama, Toru, Ahmed, Shamim, Kragh-Hansen, Otagiri, Masaki
Formato: Artigo
Idioma:Inglês
Publicado em: Springer-Verlag 2015
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2784823/
https://ncbi.nlm.nih.gov/pubmed/14727845
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1208/pt010212
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