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Amitriptyline Activates Cardiac Ryanodine Channels and Causes Spontaneous Sarcoplasmic Reticulum Calcium Release

Patients taking amitriptyline (AMT) have an increased risk of sudden cardiac death, yet the mechanism for AMT's proarrhythmic effects remains incompletely understood. Here, we hypothesize that AMT activates cardiac ryanodine channels (RyR2), causing premature Ca(2+) release from the sarcoplasmi...

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Bibliografiset tiedot
Päätekijät: Chopra, Nagesh, Laver, Derek, Davies, Sean S., Knollmann, Björn C.
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: American Society for Pharmacology and Experimental Therapeutics 2009
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC2685059/
https://ncbi.nlm.nih.gov/pubmed/18845675
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.108.051490
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