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Involvement of exon 11-associated variants of the mu opioid receptor MOR-1 in heroin, but not morphine, actions

Heroin remains a major drug of abuse and is preferred by addicts over morphine. Like morphine, heroin has high affinity and selectivity for μ-receptors, but its residual analgesia in exon 1 MOR-1 knockout mice that do not respond to morphine suggests a different mechanism of action. MOR-1 splice var...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Pan, Ying-Xian, Xu, Jin, Xu, Mingming, Rossi, Grace C., Matulonis, Joshua E., Pasternak, Gavril W.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: National Academy of Sciences 2009
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC2660730/
https://ncbi.nlm.nih.gov/pubmed/19273844
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.0811586106
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