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Synthesis and Characterization of Insulin-Transferrin Conjugates

Receptor- mediated endocytosis can be exploited for improving the transcellular delivery of therapeutic proteins. Insulin conjugated to transferrin by forming disulfide bonds has been shown to improve insulin oral bioavailability in diabetic rats. We are developing a combination strategy involving c...

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Détails bibliographiques
Auteurs principaux: Kavimandan, Nikhil J., Losi, Elena, Wilson, Jeffrey J., Brodbelt, Jennifer S., Peppas, Nicholas A.
Format: Artigo
Langue:Inglês
Publié: 2006
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC2547411/
https://ncbi.nlm.nih.gov/pubmed/17105214
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/bc050344k
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