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The synthesis and evaluation of 3-aryloxymethyl-1,2-dimethylindole-4,7-diones as mechanism-based inhibitors of NAD(P)H:quinone oxidoreductase 1 (NQO1) activity

NAD(P)H:quinone oxidoreductase 1 is a proposed target in pancreatic cancer. We describe the synthesis of a series of indolequinones, based on the 5- and 6-methoxy-1,2-dimethylindole-4,7-dione chromophores with a range of phenolic leaving groups at the (indol-3-yl)methyl position. The ability of thes...

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Detalhes bibliográficos
Main Authors: Colucci, Marie A., Reigan, Philip, Siegel, David, Chilloux, Aurélie, Ross, David, Moody, Christopher J.
Formato: Artigo
Idioma:Inglês
Publicado em: 2007
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2536657/
https://ncbi.nlm.nih.gov/pubmed/17944451
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm070396q
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