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Syntheses and optimization of new GS39783 analogues as positive allosteric modulators of GABA(B) receptors
The optimization of GS39783 into potent, selective and safe positive allosteric modulators of GABA(B) receptors is presented.
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| Glavni autori: | , , , |
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| Format: | Artigo |
| Jezik: | Inglês |
| Izdano: |
2007
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| Teme: | |
| Online pristup: | https://ncbi.nlm.nih.gov/pmc/articles/PMC2278029/ https://ncbi.nlm.nih.gov/pubmed/17884493 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2007.09.023 |
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