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Pharmacological activity of (-)-discretamine, a novel vascular alpha-adrenoceptor and 5-hydroxytryptamine receptor antagonist, isolated from Fissistigma glaucescens.

1. The pharmacological activity of (-)-discretamine, isolated from Fissistigma glaucescens, was determined in rat isolated thoracic aorta, cardiac tissues and ventricular myocytes and guinea-pig isolated trachea. 2. (-)-Discretamine was found to be an alpha 1-adrenoceptor blocking agent in rat thora...

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Autori principali: Ko, F. N., Yu, S. M., Su, M. J., Wu, Y. C., Teng, C. M.
Natura: Artigo
Lingua:Inglês
Pubblicazione: Nature Publishing Group 1993
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2175899/
https://ncbi.nlm.nih.gov/pubmed/7902181
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