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Solubilization and characterization of GABAB receptor binding sites from porcine brain synaptic membranes.

1. The characteristics of membrane bound GABAB receptors in pig brain are similar to those in rat brain as judged by in vitro binding experiments and sensitivity to GTP. The rank order of affinity of GABAB receptor ligands was CGP 54626 > GABA approximately (-)-baclofen >> CGP 35348 = CGP 3...

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Detalles Bibliográficos
Main Authors: Facklam, M., Bowery, N. G.
Formato: Artigo
Idioma:Inglês
Publicado: Nature Publishing Group 1993
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC2175871/
https://ncbi.nlm.nih.gov/pubmed/8306067
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