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Antagonist effects of seglitide (MK 678) at somatostatin receptors in guinea-pig isolated right atria.

Somatostatin (SS) exerts a negative inotropic effect in isolated atria. Here we report that in guinea-pig isolated right atria, seglitide, a potent cyclic hexapeptide somatostatin agonist, behaves as a competitive somatostatin receptor antagonist with pA2 values against SS14, SS25 and SS28, of 6.50...

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Autores principales: Dimech, J., Feniuk, W., Humphrey, P. P.
Formato: Artigo
Lenguaje:Inglês
Publicado: Nature Publishing Group 1993
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC2175736/
https://ncbi.nlm.nih.gov/pubmed/8104651
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