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Identification of benzomorphan-kappa opiate receptors in cerebral arteries which subserve relaxation.

Several 'so-called' kappa-opiate receptor agonists e.g., ketocyclazocine (Kc), ethylketocyclazocine (Ekc), bremazocine, MR-2034 and U-50488H, were tested on basilar and middle cerebral arteries of the dog in vitro for relaxant or contractile activities. Ekc, Kc and bremazocine were found t...

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Autori principali: Altura, B. T., Altura, B. M., Quirion, R.
Natura: Artigo
Lingua:Inglês
Pubblicazione: Nature Publishing Group 1984
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC1987038/
https://ncbi.nlm.nih.gov/pubmed/6329394
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