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A novel series of non-quaternary oxadiazoles acting as full agonists at muscarinic receptors

1 A novel series of non-quaternary oxadiazole-based muscarinic agonists demonstrated high affinity for muscarinic receptors. 2 These agonists possessed high efficacy in the nanomolar range at muscarinic receptors in the superior cervical ganglion, atrium and ileum but did not show selectivity across...

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Main Authors: Freedman, S.B., Harley, E.A., Patel, S., Newberry, N.R., Gilbert, M.J., McKnight, A.T., Tang, J.K., Maguire, J.J., Mudunkotuwa, N.T., Baker, R., Street, L.J., MacLeod, A.M., Saunders, J., Iversen, L.L.
Formato: Artigo
Idioma:Inglês
Publicado em: 1990
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC1917727/
https://ncbi.nlm.nih.gov/pubmed/2076477
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