Failure of BQ123, a more potent antagonist of sarafotoxin 6b than of endothelin-1, to distinguish between these agonists in binding experiments.

Lignende værker

• Characterization of the endothelin receptor selective agonist, BQ3020 and antagonists BQ123, FR139317, BQ788, 50235, Ro462005 and bosentan in the heart.
  af: Peter, M. G., et al.
  Udgivet: (1996)
• Dose- and time-dependency of the dilator effects of the endothelin antagonist, BQ-123, in the human forearm
  af: Berrazueta, José R., et al.
  Udgivet: (1997)
• Reversal of established responses to endothelin-1 in vivo and in vitro by the endothelin receptor antagonists, BQ-123 and PD 145065.
  af: Warner, T. D., et al.
  Udgivet: (1994)
• Endothelins are more sensitive than sarafotoxins to neutral endopeptidase: possible physiological significance.
  af: Skolovsky, M, et al.
  Udgivet: (1990)
• Early therapeutic experience with the endothelin antagonist BQ-123 in pulmonary hypertension after congenital heart surgery
  af: Prendergast, B, et al.
  Udgivet: (1999)