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Pharmacological profile of GR117289 in vitro: a novel, potent and specific non-peptide angiotensin AT1 receptor antagonist.

1. This paper describes the effects of GR117289 (1-[[3-bromo-2-[2-(1H-tetrazol-5-yl)phenyl]-5-benzo-furanyl]methyl ]-2-butyl-4-chloro-1H-imidazole-5-carboxylic acid) at angiotensin receptors and binding sites in rabbit aorta, rat liver and bovine cerebellum preparations in vitro. 2. In rabbit isolat...

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Autores principales: Robertson, M. J., Barnes, J. C., Drew, G. M., Clark, K. L., Marshall, F. H., Michel, A., Middlemiss, D., Ross, B. C., Scopes, D., Dowle, M. D.
Formato: Artigo
Lenguaje:Inglês
Publicado: 1992
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC1907952/
https://ncbi.nlm.nih.gov/pubmed/1467838
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