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Computational screening of inhibitors for HIV-1 integrase using a receptor based pharmacophore model

The HIV (human immuno­deficiency virus) integrase has a crucial role in viral replication. Moreover, it has no cellular homologue in humans. Hence, it is considered as an attractive drug target. Many inhibitors against the integrase protein has been designed and discussed. The Y-3 inhibitor (4-acety...

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Detalhes bibliográficos
Main Authors: Jaganatharaja, Janani, Gowthaman, Ragul
Formato: Artigo
Idioma:Inglês
Publicado em: Biomedical Informatics Publishing Group 2006
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC1891665/
https://ncbi.nlm.nih.gov/pubmed/17597868
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