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U-90152, a potent inhibitor of human immunodeficiency virus type 1 replication.

Bisheteroarylpiperazines are potent inhibitors of human immunodeficiency virus type 1 (HIV-1) reverse transcriptase (RT). We describe a novel bisheteroarylpiperazine, U-90152 [1-(5-methanesulfonamido-1H-indol-2-yl-carbonyl)-4-[3-(1-methyl eth yl-amino)pyridinyl]piperazine], which inhibited recombina...

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Main Authors: Dueweke, T J, Poppe, S M, Romero, D L, Swaney, S M, So, A G, Downey, K M, Althaus, I W, Reusser, F, Busso, M, Resnick, L
Formato: Artigo
Idioma:Inglês
Publicado: 1993
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC187915/
https://ncbi.nlm.nih.gov/pubmed/7685995
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