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Interference of transcriptional activation by the antineoplastic drug ecteinascidin-743

Ecteinascidin-743 (ET-743) is a tetrahydroisoquinoline alkaloid isolated from the tunicate Ecteinascidia turbinata currently under phase II clinical trials for its potent anticancer activity. ET-743 binds DNA in the minor groove and forms covalent adducts with some sequence specificity. It selective...

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Main Authors: Minuzzo, Mario, Marchini, Sergio, Broggini, Massimo, Faircloth, Glynn, D'Incalci, Maurizio, Mantovani, Roberto
Formato: Artigo
Idioma:Inglês
Publicado: National Academy of Sciences 2000
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC18737/
https://ncbi.nlm.nih.gov/pubmed/10841573
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