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Pharmacological profile of PD 117302, a selective kappa-opioid agonist.

1 PD 117302, a new nonpeptide opioid compound shown in in vitro studies to be a selective kappa-opioid agonist, has been evaluated in vivo for antinociceptive activity and other effects characteristic of kappa-receptor activation. 2 Dose-related long lasting antinociception was produced by PD 117302...

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Main Authors: Leighton, G. E., Johnson, M. A., Meecham, K. G., Hill, R. G., Hughes, J.
Formato: Artigo
Idioma:Inglês
Publicado: 1987
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC1853714/
https://ncbi.nlm.nih.gov/pubmed/2827830
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