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Evolving the lock to fit the key to create a family of G protein-coupled receptors potently activated by an inert ligand

We evolved muscarinic receptors in yeast to generate a family of G protein-coupled receptors (GPCRs) that are activated solely by a pharmacologically inert drug-like and bioavailable compound (clozapine-N-oxide). Subsequent screening in human cell lines facilitated the creation of a family of muscar...

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Détails bibliographiques
Auteurs principaux: Armbruster, Blaine N., Li, Xiang, Pausch, Mark H., Herlitze, Stefan, Roth, Bryan L.
Format: Artigo
Langue:Inglês
Publié: National Academy of Sciences 2007
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC1829280/
https://ncbi.nlm.nih.gov/pubmed/17360345
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.0700293104
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