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Suc-[Glu(9), Ala(11,15)]-endothelin-1 (8–21), IRL 1620, identifies two populations of ET(B) receptors in guinea-pig bronchus

1. The pharmacological properties of endothelin receptors (ETR) were investigated in guinea-pig bronchus by comparing binding and functional results. 2. In binding assays, both the ET(B) agonists, endothelin-3 (ET-3) and N-suc-[Glu(9),Ala(11,15)]ET-1(8–21) (IRL 1620), and the antagonist, N-cis-2,6-d...

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Autors principals: Mazzoni, Maria R, Breschi, M Cristina, Ceccarelli, Francesca, Lazzeri, Nicola, Giusti, Laura, Nieri, Paola, Lucacchini, Antonio
Format: Artigo
Idioma:Inglês
Publicat: 1999
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC1760658/
https://ncbi.nlm.nih.gov/pubmed/10455290
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0702672
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