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The general anesthetic propofol increases brain N-arachidonylethanolamine (anandamide) content and inhibits fatty acid amide hydrolase

1. Propofol (2,6-diisopropylphenol) is widely used as a general anesthetic and for the maintenance of long-term sedation. We have tested the hypothesis that propofol alters endocannabinoid brain content and that this effect contributes to its sedative properties. 2. A sedating dose of propofol in mi...

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Autors principals: Patel, Sachin, Wohlfeil, Eric R, Rademacher, David J, Carrier, Erica J, Perry, LaToya J, Kundu, Abhijit, Falck, J R, Nithipatikom, Kasem, Campbell, William B, Hillard, Cecilia J
Format: Artigo
Idioma:Inglês
Publicat: 2003
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC1573928/
https://ncbi.nlm.nih.gov/pubmed/12839875
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0705334
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