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Effect of sildenafil on cyclic nucleotide phosphodiesterase activity, vascular tone and calcium signaling in rat pulmonary artery

1. Sildenafil (viagra) is a potent PDE5 inhibitor and thus a relaxant drug in corpus carvernosum smooth muscle. In the present work, we evidenced the presence of PDE5 isozyme and investigated the effect of sildenafil on the specific cyclic nucleotide phosphodiesterase (PDE) activity, smooth muscle t...

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Autores principales: Pauvert, O, Lugnier, C, Keravis, T, Marthan, R, Rousseau, E, Savineau, J P
Formato: Artigo
Lenguaje:Inglês
Publicado: 2003
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC1573876/
https://ncbi.nlm.nih.gov/pubmed/12788811
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0705277
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