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Activation of vanilloid receptor 1 by resiniferatoxin mobilizes calcium from inositol 1,4,5-trisphosphate-sensitive stores

1. Capsaicin and resiniferatoxin (RTX) stimulate Ca(2+) influx by activating vanilloid receptor 1 (VR1), a ligand-gated Ca(2+) channel on sensory neurones. We investigated whether VR1 activation could also trigger Ca(2+) mobilization from intracellular Ca(2+) stores. 2. Human VR1-transfected HEK293...

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Detalhes bibliográficos
Main Authors: Marshall, Ian C B, Owen, Davina E, Cripps, Tim V, Davis, John B, McNulty, Shaun, Smart, Darren
Formato: Artigo
Idioma:Inglês
Publicado em: 2003
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC1573630/
https://ncbi.nlm.nih.gov/pubmed/12522087
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0705003
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