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α(1B) adrenergic receptors in gonadotrophin-releasing hormone neurones: relation to Transport-P

1. Peptidergic neurones accumulate amines via an unusual uptake process, designated Transport-P. [(3)H]-prazosin binds to α(1) adrenoceptors on these cells and is displaceable by unlabelled prazosin in concentrations up to 10(−7) M. However, at greater concentrations of prazosin, there is a paradoxi...

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Autors principals: Al-Damluji, S, Shen, W B, White, S, Barnard, E A
Format: Artigo
Idioma:Inglês
Publicat: 2001
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC1572539/
https://ncbi.nlm.nih.gov/pubmed/11156594
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0703781
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