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Inhibition of NFκB-mediated pro-inflammatory gene expression in rat mesangial cells by the enolized 1,3-dioxane-4,6-dione-5-carboxamide, CGP-43182

1. CGP-43182 has been described as a potent inhibitor of group IIA secreted phospholipase A(2) (group IIA sPLA(2)) activity in vitro. In rat mesangial cells, inhibition of group IIA sPLA(2) activity by CGP-43182 results in a 70% reduction of cytokine-stimulated prostaglandin E(2) biosynthesis, sugge...

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Autors principals: Scholz-Pedretti, Kirsten, Eberhardt, Wolfgang, Rupprecht, Gerhard, Beck, Karl-Friedrich, Spitzer, Silke, Pfeilschifter, Josef, Kaszkin, Marietta
Format: Artigo
Idioma:Inglês
Publicat: 2000
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC1572174/
https://ncbi.nlm.nih.gov/pubmed/10882405
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0703419
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