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Compounds that block both intermediate-conductance (IK(Ca)) and small-conductance (SK(Ca)) calcium-activated potassium channels

1. Nine bis-quinolinyl and bis-quinolinium compounds related to dequalinium, and previously shown to block apamin-sensitive small conductance Ca(2+)-activated K(+) channels (SK(Ca)), have been tested for their inhibitory effects on actions mediated by intermediate conductance Ca(2+)-activated K(+) c...

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Autores principales: Malik-Hall, M, Ganellin, C R, Galanakis, D, Jenkinson, D H
Formato: Artigo
Lenguaje:Inglês
Publicado: 2000
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC1571984/
https://ncbi.nlm.nih.gov/pubmed/10742299
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0703233
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