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Block of gating currents related to K(+) channels as a mechanism of action of clofilium and d-sotalol in isolated guinea-pig ventricular heart cells

1. The possibility that the class III antiarrhythmic drugs clofilium and d-sotalol might affect delayed rectifier potassium channels at the level of their gating currents was assessed with the whole-cell patch-clamp technique in guinea-pig isolated ventricular heart cells. 2. Clofilium (up to 20 μM)...

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Autori principali: Malécot, Claire O, Argibay, Jorge A
Natura: Artigo
Lingua:Inglês
Pubblicazione: 1999
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC1571629/
https://ncbi.nlm.nih.gov/pubmed/10510439
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/sj.bjp.0702768
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