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Effects of cyclothiazide on GluR1/AMPA receptors

Cyclothiazide (CTZ), a positive allosteric modulator of ionotropic α-amino-3-hydroxy-5-methylisoxazole-4-propionic acid (AMPA)-type glutamate receptors, is used frequently to block the desensitization of both native and heterologously expressed AMPA receptors. Specifically, CTZ is known to produce a...

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Autors principals: Fucile, Sergio, Miledi, Ricardo, Eusebi, Fabrizio
Format: Artigo
Idioma:Inglês
Publicat: National Academy of Sciences 2006
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC1413821/
https://ncbi.nlm.nih.gov/pubmed/16473938
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.0511063103
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