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Crystal structure of NS-134 in complex with bovine cathepsin B: a two-headed epoxysuccinyl inhibitor extends along the entire active-site cleft

The crystal structure of the inhibitor NS-134 in complex with bovine cathepsin B reveals that functional groups attached to both sides of the epoxysuccinyl reactive group bind to the part of active-site cleft as predicted. The -Leu-Pro-OH side binds to the primed binding sites interacting with the H...

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Bibliografiska uppgifter
Huvudupphovsmän: Štern, Igor, Schaschke, Norbert, Moroder, Luis, Turk, Dušan
Materialtyp: Artigo
Språk:Inglês
Publicerad: Portland Press Ltd. 2004
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Länkar:https://ncbi.nlm.nih.gov/pmc/articles/PMC1133859/
https://ncbi.nlm.nih.gov/pubmed/15084146
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1042/BJ20040237
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