Stereoselective synthesis of fused tetrahydroquinazolines through one-pot double [3 + 2] dipolar cycloadditions followed by [5 + 1] annulation

The one-pot [3 + 2] cycloaddition of an azomethine ylide with a maleimide followed by another [3 + 2] cycloaddition of an azide with the second maleimide gives a 1,5-diamino intermediate which is used for a sequential aminomethylation reaction with formaldehyde through [5 + 1] annulation to afford a...

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Ngā kaituhi matua:	Xiaofeng Zhang, Kenny Pham, Shuai Liu, Marc Legris, Alex Muthengi, Jerry P. Jasinski, Wei Zhang
Hōputu:	Artigo
Reo:	Inglês
I whakaputaina:	Beilstein-Institut 2016-10-01
Rangatū:	Beilstein Journal of Organic Chemistry
Ngā marau:	[5 + 1] annulation [3 + 2] cycloaddition one-pot reactions stereoselective synthesis tetrahydroquinazoline
Urunga tuihono:	https://doi.org/10.3762/bjoc.12.211
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