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Inhibition Analysis and High-Resolution Crystal Structure of <i>Mus musculus</i> Glutathione Transferase P1-1

Multidrug resistance is a significant barrier that makes anticancer therapies less effective. Glutathione transferases (GSTs) are involved in multidrug resistance mechanisms and play a significant part in the metabolism of alkylating anticancer drugs. The purpose of this study was to screen and sele...

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Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Oleksii Kupreienko, Fotini Pouliou, Konstantinos Konstandinidis, Irene Axarli, Eleni Douni, Anastassios C. Papageorgiou, Nikolaos E. Labrou
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: MDPI AG 2023-03-01
Saila:Biomolecules
Gaiak:
Sarrera elektronikoa:https://www.mdpi.com/2218-273X/13/4/613
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