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Impact of Crystal Habit on the Dissolution Rate and In Vivo Pharmacokinetics of Sorafenib Tosylate

The dissolution rate is the rate-limiting step for Biopharmaceutics Classification System (BCS) class II drugs to enhance their in vivo pharmacokinetic behaviors. There are some factors affecting the dissolution rate, such as polymorphism, particle size, and crystal habit. In this study, to improve...

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Bibliografski detalji
Glavni autori: Chi Uyen Phan, Jie Shen, Kaxi Yu, Jianming Mao, Guping Tang
Format: Artigo
Jezik:Inglês
Izdano: MDPI AG 2021-06-01
Serija:Molecules
Teme:
Online pristup:https://www.mdpi.com/1420-3049/26/11/3469
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