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Inhibitory effect of clemastine on P-glycoprotein expression and function: an in vitro and in situ study

Objective(s):Transporters have an important role in pharmacokinetics of drugs. Inhibition or induction of drug transporters activity can affect drug absorption, safety, and efficacy. P-glycoprotein (P-gp) is the most important membrane transporter that is responsible for active efflux of drugs. It i...

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Principais autores: Mehran Mesgari Abbasi, Hadi Valizadeh, Hamed Hamishekar, Leila Mohammadnejad, Parvin Zakeri-Milani
Formato: Artigo
Idioma:Inglês
Publicado em: Mashhad University of Medical Sciences 2016-04-01
coleção:Iranian Journal of Basic Medical Sciences
Assuntos:
Acesso em linha:http://ijbms.mums.ac.ir/article_6815_563c9975ba66430234720970c3946166.pdf
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