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The Evaluation of (1<i>R</i>,4<i>R</i>,7<i>R</i>,10<i>R</i>)-α,α′,α″,α‴-Tetramethyl-1,4,7,10-tetraazacyclododecane-1,4,7,10-tetraacetic Acid (DOTMA) as a Chelator for Zirconium-89

Recently, macrocycles such as 1,4,7,10-tetraazacyclododecane-1,4,7,10-tetraacetic acid (DOTA) have been observed to form zirconium-89 (<sup>89</sup>Zr: t<sub>½</sub> = 78.4 h, β+: 22.8%, E<sub>β+max</sub> = 901 keV; EC: 77%, E<sub>γ</sub> = 909 keV)-complexes with excellent in vivo stability. In thi...

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Autori principali: Darpan N. Pandya, Pere Miro, Michael A. Sinnwell, George B. Crull, Thaddeus J. Wadas
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI AG 2025-10-01
Serie:Molecules
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Accesso online:https://www.mdpi.com/1420-3049/30/20/4129
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