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Opportunities for protein kinase drug discovery – 2025 update on the chemically underexplored human kinome

As a part of the Illuminating the Druggable Genome initiative, the U.S. National Institutes of Health (NIH), identified 162 understudied human protein and lipid kinases forming the “dark” kinome. In protein kinase (PK) drug discovery, the dark kinome has become a focal point in the search for new PK...

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Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Selina Koch, Elena Kullmann, Jürgen Bajorath
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: Elsevier 2025-12-01
Saila:European Journal of Medicinal Chemistry Reports
Gaiak:
Sarrera elektronikoa:http://www.sciencedirect.com/science/article/pii/S2772417425000615
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