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Structure-guided discovery of novel dUTPase inhibitors with anti-Nocardia activity by computational design

The zoonosis caused by Nocardia is increasing seriously. But commonly used antibiotic drugs often lead to resistance. N. seriolae dUTPase (NsdUTPase) plays a key role in the proliferation of Nocardia, and was regarded as a potent drug target. However, there was little report about the NsdUTPase inhi...

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Autori principali: Zhi-Zheng Wang, Jun Weng, Jing Qi, Xin-Xin Fu, Ban-Bin Xing, Yang Hu, Chun-Hsiang Huang, Chin-Yu Chen, Zigong Wei
Natura: Artigo
Lingua:Inglês
Pubblicazione: Taylor & Francis Group 2024-12-01
Serie:Journal of Enzyme Inhibition and Medicinal Chemistry
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Accesso online:https://www.tandfonline.com/doi/10.1080/14756366.2024.2411573
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